Re: COND LAPLACE LIKELIHOOD

From: Leonid Gibiansky Date: August 04, 2009 technical Source: mail-archive.com
something is incorrect here, either model or comments: P0 = C0/(1+C0) ; Probability of Score=>0 P1 = C1/(1+C1) ; Probability of Score=>1 P2 = C2/(1+C2) ; Probability of Score=>2 Probability of Score=>0 is always 1 (because score is 0 or positive number as I can see). My guess is that the model is incorrect, it should be (assuming that the drug increases probability of higher scores while natural state favors score 0) > A1 = B1 + DRUG > A2 = B1 - B2 + DRUG > A3 = B1 - B2 - B3 + DRUG > C1 = EXP(A1) > C2 = EXP(A2) > C3 = EXP(A3) > P1 = C1/(1+C1) ; Probability of Score=>1 > P2 = C2/(1+C2) ; Probability of Score=>2 > P3 = C3/(1+C3) ; Probability of Score=>3 > > PR0 = 1-P1 ; Probability of Score=0 > PR1 = P1-P2 ; Probability of Score=1 > PR2 = P2-P3 ; Probability of Score=2 > PR3 = P3 ; Probability of Score=3 > IF (DV.EQ.0) Y=PR0 > IF (DV.EQ.1) Y=PR1 > IF (DV.EQ.2) Y=PR2 > IF (DV.EQ.3) Y=PR3 B2 and B3 should be positive -------------------------------------- Leonid Gibiansky, Ph.D. President, QuantPharm LLC web: www.quantpharm.com e-mail: LGibiansky at quantpharm.com tel: (301) 767 5566 [email protected] wrote: > Hi Samer, > Thanks for your quick reply. Here is my control stream: > > $SUBS ADVAN6 TOL=6 > $MODEL > COMP=(ABSO) > COMP=(CENT) > COMP=(PERI) > COMP=(EFFECT) > $PK > CL =ICL*24 > V2 = IVC > Q=... > K23=Q/V2 > V3= > K32=Q/V3 > K=CL/V2 > KA=... > KE0 = THETA(6) > B1 = THETA(1) > B2 = THETA(2) > B3 = THETA(3) > EMAX = THETA(4) > EC50 = THETA(5)*EXP(ETA(1)) > > $DES > DADT(1)=-A(1)*KA > DADT(2)=A(1)*KA-A(2)*K23+A(3)*K32-A(2)*K > DADT(3)=A(2)*K23-A(3)*K32 > DADT(4)=KE0*(A(2)/V2-A(4)) > > $ERROR > CE=A(4) > DRUG = EMAX*CE/(EC50+CE) > A0 = B1 + DRUG > A1 = B1 + B2 + DRUG > A2 = B1 + B2 + B3 + DRUG > C0 = EXP(A0) > C1 = EXP(A1) > C2 = EXP(A2) > P0 = C0/(1+C0) ; Probability of Score=>0 > P1 = C1/(1+C1) ; Probability of Score=>1 > P2 = C2/(1+C2) ; Probability of Score=>2 > > PR0 = P0 ; Probability of Score=0 > PR1 = P1-P0 ; Probability of Score=1 > PR2 = P2-P1 ; Probability of Score=2 > PR3 = 1-P2 ; Probability of Score=3 > IF (DV.EQ.0) Y=PR0 > IF (DV.EQ.1) Y=PR1 > IF (DV.EQ.2) Y=PR2 > IF (DV.EQ.3) Y=PR3 > > $THETA (-20 -6.3) ; THETA1 B1 > $THETA (-10 -0.3) ; THETA2 B2 > $THETA (-10 2) ; THETA3 B3 > $THETA (0 5) ; THETA4 EMAX > $THETA (0 50) ; THETA5 EC50 > $THETA (0 1) ; THETA6 KEO > > $OMEGA 2 > > $ESTIMATION MAXEVAL=9999 PRINT=5 METHOD=COND LAPLACIAN LIKELIHOOD NOABORT MSFO=MSF1 Here I include the dataset for first two subjects. Since it is a simultaneous PKPD link model, DV in the data set as follows is categorical PD data. The dose was given daily and DV was recorded daily as well. > > #SUBJ TIME AMT EVID II ADDL PD KA CL V2 MDV > 1 0 . 0 . . 0 9.96 4.12 63.57 0 > 1 0 1 1 1 20 . 9.96 4.12 63.57 1 > 1 1 . 0 . . 0 9.96 4.12 63.57 0 > 1 2 . 0 . . 0 9.96 4.12 63.57 0 > 1 3 . 0 . . 0 9.96 4.12 63.57 0 > 1 4 . 0 . . 0 9.96 4.12 63.57 0 > 1 5 . 0 . . 0 9.96 4.12 63.57 0 > 1 6 . 0 . . 0 9.96 4.12 63.57 0 > 1 7 . 0 . . 0 9.96 4.12 63.57 0 > 1 8 . 0 . . 0 9.96 4.12 63.57 0 > 1 9 . 0 . . 0 9.96 4.12 63.57 0 > 1 10 . 0 . . 0 9.96 4.12 63.57 0 > 1 11 . 0 . . 0 9.96 4.12 63.57 0 > 1 12 . 0 . . 0 9.96 4.12 63.57 0 > 1 13 . 0 . . 0 9.96 4.12 63.57 0 > 1 14 . 0 . . 0 9.96 4.12 63.57 0 > 1 15 . 0 . . 0 9.96 4.12 63.57 0 > 1 16 . 0 . . 0 9.96 4.12 63.57 0 > 1 17 . 0 . . 0 9.96 4.12 63.57 0 > 1 18 . 0 . . 0 9.96 4.12 63.57 0 > 1 19 . 0 . . 0 9.96 4.12 63.57 0 > 1 20 . 0 . . 0 9.96 4.12 63.57 0 > 1 21 . 0 . . 0 9.96 4.12 63.57 0 > 1 22 . 0 . . 0 9.96 4.12 63.57 0 > 1 23 . 0 . . 0 9.96 4.12 63.57 0 > 1 24 . 0 . . 0 9.96 4.12 63.57 0 > 1 25 . 0 . . 0 9.96 4.12 63.57 0 > 1 26 . 0 . . 0 9.96 4.12 63.57 0 > 1 27 . 0 . . 0 9.96 4.12 63.57 0 > 2 0 . 0 . . 0 1.52 4.68 66.91 0 > 2 0 2 1 1 20 . 1.52 4.68 66.91 1 > 2 1 . 0 . . 0 1.52 4.68 66.91 0 > 2 2 . 0 . . 0 1.52 4.68 66.91 0 > 2 3 . 0 . . 0 1.52 4.68 66.91 0 > 2 4 . 0 . . 0 1.52 4.68 66.91 0 > 2 5 . 0 . . 0 1.52 4.68 66.91 0 > 2 6 . 0 . . 0 1.52 4.68 66.91 0 > 2 7 . 0 . . 0 1.52 4.68 66.91 0 > 2 8 . 0 . . 0 1.52 4.68 66.91 0 > 2 9 . 0 . . 0 1.52 4.68 66.91 0 > 2 10 . 0 . . 0 1.52 4.68 66.91 0 > 2 11 . 0 . . 0 1.52 4.68 66.91 0 > 2 12 . 0 . . 1 1.52 4.68 66.91 0 > 2 13 . 0 . . 1 1.52 4.68 66.91 0 > 2 14 . 0 . . 1 1.52 4.68 66.91 0 > 2 15 . 0 . . 1 1.52 4.68 66.91 0 > 2 16 . 0 . . 1 1.52 4.68 66.91 0 > 2 17 . 0 . . 1 1.52 4.68 66.91 0 > 2 18 . 0 . . 1 1.52 4.68 66.91 0 > 2 19 . 0 . . 1 1.52 4.68 66.91 0 > 2 20 . 0 . . 1 1.52 4.68 66.91 0 > 2 21 . 0 . . 3 1.52 4.68 66.91 0 > 2 22 . 0 . . 3 1.52 4.68 66.91 0 > 2 23 . 0 . . 3 1.52 4.68 66.91 0 > 2 24 . 0 . . 3 1.52 4.68 66.91 0 > 2 25 . 0 . . 3 1.52 4.68 66.91 0 > 2 26 . 0 . . 3 1.52 4.68 66.91 0 > 2 27 . 0 . . 3 1.52 4.68 66.91 0 > 2 28 . 0 . . 2 1.52 4.68 66.91 0 > > Thanks, > Tianli > > ****************************************************************************** > > Tianli Wang > University of Minnesota, > Department of Pharmaceutics >
Quoted reply history
> On Aug 4 2009, Samer Mouksassi wrote: > > > Can you include your control (or at least your $EST bloc) > > And the proportional odds PD data. The likelihood may go wild if some > > categories are very rare or non esistent. You need to gard against over > > or underflow. > > > > -----Original Message----- > > From: [email protected] [mailto:[email protected]] > > On Behalf Of [email protected] > > Sent: 2009-08-04 13:38 > > To: NMUSERS > > Subject: [NMusers] COND LAPLACE LIKELIHOOD > > > > Dear nmusers, > > > > Has anybody seen the following error message from NONMEM: > > "CONDITIONAL LIKELIHOOD SET TO NEGATIVE VALUE > > WITH INDIVIDUAL 2 (IN INDIVIDUAL RECORD ORDERING), DATA RECORD 13"? > > What does it mean? > > > > I am trying to use conditional lapalacian likelihood method to generate > > a proportional odds model dealing with categorical PD data. Here is a > > little piece of my data set: > > SUBJ TIME AMT EVID II ADDL DV CL V > > MDV > > 2 0 . 0 . . 0 4.12 63 > > 0 > > 2 0 1 1 1 20 . 4.12 63 > > 1 > > 2 0.005 . 2 . . . 4.12 63 > > 1 > > 2 0.01 . 2 . . . 4.12 63 > > 1 > > . > > . > > . > > 2 12 . 0 . . 0 4.12 63 > > 0 > > 2 13 . 0 . . 1 4.12 63 > > 0 > > . > > . > > . > > > > But I don't think the problem exists in the data set because I tried deleting the rows indicated in the error message, but the exactly same message still came out and NONMEM stopped running. I have no idea what's > > > > the problem for my model. > > > > Thanks in advance, > > > > Tianli
Aug 04, 2009 Wangx826 COND LAPLACE LIKELIHOOD
Aug 04, 2009 Leonid Gibiansky Re: COND LAPLACE LIKELIHOOD
Aug 05, 2009 Mats Karlsson RE: COND LAPLACE LIKELIHOOD