RE: PD interaction between two substances

From: William Bachman Date: April 05, 2004 technical Source: cognigencorp.com
From: Bachman, William (MYD) bachmanw@iconus.com Subject: RE: [NMusers] PD interaction between two substances Date: Mon, April 5, 2004 9:15 am Johan, Do I understand your question correctly: "how do I fit simultaneously PK and PD data simultaneously if I have two different PK observations and one PD observation?". If so, you have to structure your model so that each observation is modeled in a different compartment. Then instead of a binary switching mechanism based on the CMT data, you have to construct a switch based on three compartments. There may be some nuances I have not considered, but, basically: $ERROR ;IF CMT=1 for C(1), CMT=2 for C(2), CMT=3 for Effect C1=A(1)/V1 C2=A(2)/V2 IF (CT.EQ.3) THEN Y=Emax *(1/(1 + EC51/C1)* (1 + C2/EC52) + 1/(1 + EC52)/(C2) * (1 + C1/EC51)) + ERR(3) ELSEIF (CMT.EQ.1) THEN Y =F*EXP(ERR(1)) ;F is pred in CMT 1 here ELSE Y =F*EXP(ERR(2)) ;F is pred in CMT 2 here ENDIF ;check for typos in above Bill William J. Bachman, Ph.D. Manager, Pharmacometrics Research and Development GloboMax The Strategic Pharmaceutical Development Division of ICON plc 7250 Parkway Drive, Suite 430 Hanover, MD 21076 410-782-2212 bachmanw@iconus.com
Apr 05, 2004 Johan Rosenborg PD interaction between two substances
Apr 05, 2004 William Bachman RE: PD interaction between two substances
Apr 05, 2004 Immanuel Freedman RE: : PD interaction between two substances